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Search Result

Search Results for " a-1 protease inhibitor "

Targets

SARS-CoV HIV Protease

130

Compounds

14

Natural Products

1884

Recombinant Proteins

1

Libraries

3

Reagents

Cat No. Product Name Synonyms Targets
T4578 Tipranavir PNU-140690 SARS-CoV , HIV Protease
Tipranavir is a protease inhibitor that inhibits HIV-1 resistant to more than 1 protease inhibitor .Tipranavir effectively inhibits HIV-1 protease enzyme activity and dimerisation and has potent activity against multiple...
T80672 1,4-Dihydroxynaphthalene Naphthalene-1,4-diol HSV
1,4-Dihydroxynaphthalene A potent HSV-1 protease inhibitor with inhibitory effects on the HCMV protease, which can be used to study herpesviruses.
T13268 USP7-IN-1 DUB
USP7-IN-1 is a selective and reversible ubiquitin-specific protease 7 (USP7) inhibitor (IC50 = 77 μM).
T4338 USP7/USP47 inhibitor USP7/47 inhibitor-1 DUB
USP7/USP47 inhibitor (USP7/47 inhibitor-1) is a selective ubiquitin-specific protease 7/47 (USP7/USP47) inhibitor, with EC50s of 0.42 μM and 1.0 μM, respectively.
T9216 MLT-943 MLT943 MALT
MLT-943 is a potent, selective and orally active MALT1 protease inhibitor. [1].
T4317 PF 429242 NPC1L1 , Lipid
PF-429242 is a competitive inhibitor of sterol regulatory element-binding protein (SREBP) site 1 protease (IC50 = 0.175 μM). It is selective for site 1 protease against a panel of serine proteases. PF-429242 inhibits rat...
T1623 Lopinavir ABT-378 SARS-CoV , HIV Protease
Lopinavir (ABT-378) is a peptidomimetic HIV protease inhibitor that retains activity against HIV protease with the Val 82 mutation. Lopinavir is less affected by binding to serum proteins than the structurally-related dr...
T9458 PF-00835231 SARS-CoV
PF-00835231 is a CoV-2 cysteine 3C-like protease (3CLpro) inhibitor, with IC50s of 0.27 nM and 4 nM for SARS CoV-2 and SARS CoV-1 3CLpro, respectively.PF-00835231 is the active compound of the first anti-3CLpro regimen i...
T22168 Vialinin A Terrestrin A DUB
Vialinin A (Terrestrin A), a p-terphenyl compound, exhibits antioxidant properties and acts as a potent inhibitor of TNF-α, USP4, USP5, and sentrin/SUMO-specific protease 1 (SENP1). Its efficacy in autoimmune diseases an...
T12926 SJB3-019A Others , DUB
SJB3-019A is a potent, potent and novel ubiquitin-specific protease 1 (USP1) inhibitor, which promotes ID1 degradation and cytotoxicity in K562 cells 5 times more than SJB2-043, with IC50 of 0.0781 μM. SJB3-019A inhibits...
T24362 L 756423 L756423,MK-944a,MK944a,L-756,423,L-756423,MK 944a HIV Protease
L 756423 (L756423) is a novel potent and selective and competitive HIV protease inhibitor with a Ki value of 0.049 nM for HIV-1 PR.L 756423 blocks the spread of HIV(IIIb)-infected MT25 lymphocytes at 0.50-0.1 nM and can ...
T3226 Paritaprevir ABT-450,Veruprevir HCV Protease
Paritaprevir (ABT-450) is an orally bioavailable, synthetic acylsulfonamide inhibitor of the hepatitis C virus (HCV) protease complex comprised of non-structural protein 3 and 4A (NS3/NS4A), with potential activity again...
T37173 MPro Inhibitor 11a
MProinhibitor 11a is an inhibitor of severe acute respiratory syndrome coronavirus 2 (SARS-CoV-2) main protease (MPro; IC50= 0.053 μM in a TR-FRET assay).1It reduces viral yield in the culture supernatant of SARS-CoV-2-i...
T9574 PF-07304814 Lufotrelvir
Lufotrelvir (PF-07304814) is a phosphate prodrug of PF-00835231 which acts as a potent 3CL pro protease ( M pro ) inhibitor with SARS-CoV-2 antiviral activity. Lufotrelvir binds and inhibits SARS-CoV-2 3CL pro activity w...
T36682 USP30 inhibitor 18 DUB
USP30 inhibitor 18 is a selective USP30 inhibitor with an IC50 of 0.02 μM. USP30 inhibitor 18 increases protein ubiquitination and accelerates mitophagy[1]. [1]. Arthur F Kluge, et al. Novel highly selective inhibitors o...
T26446 A 77003 A-77003,Abbott 77003,A77003
A 77003 is a HIV-1 protease inhibitor. A77003 impairs HIV-1 protease-mediated Gag processing.
T26445 A 76889 A76889,A-76889
A 76889 is an inhibitor of HIV-1 protease.
T26451 A 80987 A80987,A-80987
A 80987 is an inhibitor of HIV-1 protease.
T15683 L-689502 HIV Protease
L-689502 is a potent HIV-l protease inhibitor (IC50: 1 nM).
T70518 CGP-53437
CGP-53437 is a novel HIV-1 protease inhibitor, also potently inhibiting major aspartyl peptidase 1 (May1), a secreted Cryptococcus neoformans protease.
T24266 KNI-1657
KNI-1657 is a potent and selective HIV-1 protease inhibitor (Anti-HIV-1 pNL4-3, EC50: 3 nM). KNI-1657 is a highly potent HIV-1 Protease Inhibitor against Lopinavir.
T36306 FT206
FT206 is a carboxamide inhibitor of ubiquitin-specific protease[1].
T24737 Rpi 856 A Rpi856 A,Rpi 856 B,Rpi-856 A,Rpi-856 B,Rpi856 B
Rpi 856 A is a retrovirus protease inhibitor. It is effective against HIV-1 and HTLV-1 proteases.
T30839 Cgp 53820 Cgp53820,Cgp-53820
CGP 53820 is a pseudosymmetric inhibitor of HIV-1 Protease.
T24008 DMP 323 JCR424,DMP-323,JCR-424,JCR 424,DMP323
DMP 323 is a potent inhibitor of HIV-1 protease.
T13417 ZYZ-488 Others
ZYZ-488 is a competitive inhibitor of apoptotic protease activating factor-1 (Apaf-1).
T26440 A 74704 A-74704,A74704
A 74704 is a pseudo C2-symmetric inhibitor of HIV-1 protease and its diester analog.
T26128 Rpi 856 C Rpi-856 C,Rpi856 C,Rpi-856 D,Rpi856 D,Rpi 856 D
Rpi 856 C is a retrovirus protease inhibitor from Streptomyces that is effective against HIV-1 and HTLV-1 proteases.
T30841 Cgp 57813 Cgp-57813,Cgp57813
CGP 57813 is a lipophilic compound, which can be used as an inhibitor of HIV-1 protease.
T40068 SENP1-IN-1 SENP1-IN-1
SENP1-IN-1 is a distinct inhibitor of the deSUMOylation protease 1 (SENP1), designed to enhance tumor radiosensitivity.
T10082 DPP-IV-IN-1 Others
DPP-IV-IN-1 is an effective inhibitor of dipeptidyl peptidase IV (DPP-IV), a serine protease (IC50: 4.6 nM).
T70717 KNI 174
KNI 174 is a new type of anti‐AIDS drug used as an HIV‐1 protease inhibitor
T40067 SENP1-IN-4 SENP1-IN-4
SENP1-IN-4, a distinct inhibitor of the deSUMOylation protease 1 (SENP1), is designed to enhance tumor radiosensitivity.
T63949 HIV-1 protease-IN-2
HIV-1 protease-IN-2 is a potent inhibitor of HIV-1 protease (IC50: 2.53 nM). HIV-1 protease-IN-2 exhibits antiviral effects against DRV (Darunavir) sensitive or drug resistant HIV-1 mutants.
T40069 SENP1-IN-2 SENP1-IN-2
SENP1-IN-2, a distinct inhibitor of the deSUMOylation protease 1 (SENP1), is designed to enhance tumor radiosensitivity.
T40066 SENP1-IN-3 SENP1-IN-3
SENP1-IN-3 is a distinct inhibitor of the deSUMOylation protease 1 (SENP1), designed to enhance tumor radiosensitivity.
T8675 Vaniprevir Others
Vaniprevir is a macrocyclic hepatitis C virus NS3/4a protease inhibitor and is active against both the genotype 1 and genotype 2 NS3/4a protease enzymes. vaniprevir has good plasma exposure and excellent liver exposure...
T30585 Brecanavir GW-640385,GW-640385X,UNII-E367I8C7FI,CHEMBL206031,GW-0385
Brecanavir is a tyrosyl-based arylsulfonamide, high affinity, protease inhibitor (PI) for the treatment of human immunodeficiency virus type 1.
T15163 DPC-681 DPH-153893 Others
DPC-681 is a potent and selective HIV protease inhibitor (IC90s: 4 to 40 nM for wild-type HIV-1).
T74939 HIV protease-IN-1
HIV protease-IN-1 (compound 1·succinate), a potent non-peptidic inhibitor of HIV protease, is utilized for AIDS research [1].
T14295 Antipain Others
Antipain is a protease inhibitor isolated from Actinomycetes. Antipain inhibits N-methyl-N'-nitro-N-nitrosoguanidine (MNNG)-induced transformation and increases chromosomal aberrations[1][2].
T28306 PD 099560 PD099560,PD-099560
PD 099560 is a non-peptide inhibitor of HIV-1 protease, a significant target enzyme in AIDS research.
T35043 Vedroprevir GS9451,GS 9451,GS-9451
Vedroprevir, also known as GS9451, is a selective hepatitis C virus (HCV) NS3 protease inhibitor in the development of the treatment of genotype 1 (GT1) HCV infection.
T63453 HIV-1 protease-IN-1
HIV-1 protease-IN-1 is a potent inhibitor of HIV-1 protease (IC50: 90 pM). HIV-1 protease-IN-1 has antiviral activity against B-HIV (EC50: 89 nM): HIV-1 protease-IN-1 was able to act on C-HIV strain ZM246 (EC50: 13.59 nM...
T14187 ALLM Calpain inhibitor II Others
ALLM (Calpain inhibitor II), a potent calpain and cathepsin protease inhibitor, not only prevents neuronal cell death but also enhances chronic neurological function following spinal cord injury (SCI)[1][2].
T70491 XM 323
XM 323 is an inhibitor of clinical isolates of HIV-1 in vitro and represents a novel class of non-peptidyl inhibitors of HIV-1 protease.
T63733 HIV-1 protease-IN-6
HIV-1 protease-IN-6 (compound 17d) is a potent inhibitor of HIV-1 protease (IC50: 21 pM, Ki: 4.7 pM). HIV-1 protease-IN-6 showed significant antiviral activity against DRV (darunavir) resistant mutants, even exceeding th...
T38931 Calpain Inhibitor-1
Calpain Inhibitor-1 (compound 36) is a highly potent and selective inhibitor of Calpain 1 (Cal1), which is a cysteine protease. It exhibits an IC50 value of 100 nM and a Ki value of 2.89 μM.
T26192 SKF-107457 SKF 107457,Ala-Ala-Phepsi(CH(OH)CH2)Gly-Val-Val-OCH3
SKF-107457 is an HIV protease type 1 inhibitor. It is a hexapeptide substrate analog with the scissile bond being replaced by a hydroxy ethylene isostere.
T79537 HIV-1 protease-IN-12 HIV Protease
HIV-1 protease-IN-12 (compound 35b) serves as a potent inhibitor of HIV-1 protease, exhibiting an IC50 value of 0.51 nM, and demonstrates efficacy against drug-resistant variant [1].

Compounds

Tipranavir
T4578
Synonym: PNU-140690
Target: SARS-CoV, HIV Protease
1,4-Dihydroxynaphthalene
T80672
Synonym: Naphthalene-1,4-diol
Target: HSV
USP7-IN-1
T13268
Synonym:
Target: DUB
USP7/USP47 inhibitor
T4338
Synonym: USP7/47 inhibitor-1
Target: DUB
MLT-943
T9216
Synonym: MLT943
Target: MALT
PF 429242
T4317
Synonym:
Target: NPC1L1, Lipid
Lopinavir
T1623
Synonym: ABT-378
Target: SARS-CoV, HIV Protease
PF-00835231
T9458
Synonym:
Target: SARS-CoV
Vialinin A
T22168
Synonym: Terrestrin A
Target: DUB
SJB3-019A
T12926
Synonym:
Target: Others, DUB
L 756423
T24362
Synonym: L756423,MK-944a,MK944a,L-756,423,L-756423,MK 944a
Target: HIV Protease
Paritaprevir
T3226
Synonym: ABT-450,Veruprevir
Target: HCV Protease
MPro Inhibitor 11a
T37173
Synonym:
Target:
PF-07304814
T9574
Synonym: Lufotrelvir
Target:
USP30 inhibitor 18
T36682
Synonym:
Target: DUB
A 77003
T26446
Synonym: A-77003,Abbott 77003,A77003
Target:
A 76889
T26445
Synonym: A76889,A-76889
Target:
A 80987
T26451
Synonym: A80987,A-80987
Target:
L-689502
T15683
Synonym:
Target: HIV Protease
CGP-53437
T70518
Synonym:
Target:
KNI-1657
T24266
Synonym:
Target:
FT206
T36306
Synonym:
Target:
Rpi 856 A
T24737
Synonym: Rpi856 A,Rpi 856 B,Rpi-856 A,Rpi-856 B,Rpi856 B
Target:
Cgp 53820
T30839
Synonym: Cgp53820,Cgp-53820
Target:
DMP 323
T24008
Synonym: JCR424,DMP-323,JCR-424,JCR 424,DMP323
Target:
ZYZ-488
T13417
Synonym:
Target: Others
A 74704
T26440
Synonym: A-74704,A74704
Target:
Rpi 856 C
T26128
Synonym: Rpi-856 C,Rpi856 C,Rpi-856 D,Rpi856 D,Rpi 856 D
Target:
Cgp 57813
T30841
Synonym: Cgp-57813,Cgp57813
Target:
SENP1-IN-1
T40068
Synonym: SENP1-IN-1
Target:
DPP-IV-IN-1
T10082
Synonym:
Target: Others
KNI 174
T70717
Synonym:
Target:
SENP1-IN-4
T40067
Synonym: SENP1-IN-4
Target:
HIV-1 protease-IN-2
T63949
Synonym:
Target:
SENP1-IN-2
T40069
Synonym: SENP1-IN-2
Target:
SENP1-IN-3
T40066
Synonym: SENP1-IN-3
Target:
Vaniprevir
T8675
Synonym:
Target: Others
Brecanavir
T30585
Synonym: GW-640385,GW-640385X,UNII-E367I8C7FI,CHEMBL206031,GW-0385
Target:
DPC-681
T15163
Synonym: DPH-153893
Target: Others
HIV protease-IN-1
T74939
Synonym:
Target:
Antipain
T14295
Synonym:
Target: Others
PD 099560
T28306
Synonym: PD099560,PD-099560
Target:
Vedroprevir
T35043
Synonym: GS9451,GS 9451,GS-9451
Target:
HIV-1 protease-IN-1
T63453
Synonym:
Target:
ALLM
T14187
Synonym: Calpain inhibitor II
Target: Others
XM 323
T70491
Synonym:
Target:
HIV-1 protease-IN-6
T63733
Synonym:
Target:
Calpain Inhibitor-1
T38931
Synonym:
Target:
SKF-107457
T26192
Synonym: SKF 107457,Ala-Ala-Phepsi(CH(OH)CH2)Gly-Val-Val-OCH3
Target:
HIV-1 protease-IN-12
T79537
Synonym:
Target: HIV Protease
1 2 3
Cat No. Product Name Synonyms Targets
T4S0181 Hinokiflavone MMP , BCL , E1/E2/E3 Enzyme
Hinokiflavone, a novel modulator of pre-mRNA splicing activity both in vitro and in cellulo, inhibits the assembly of the spliceosome, particularly blocking the formation of the B complex. Additionally, it acts as a SUMO...
TN1059 Ganoderic acid B IL Receptor , HIV Protease , JAK , STAT
Ganoderic acid B is a chemical marker in quality control of G. lucidum and related products. Ganoderic acid B-containing herbs has potential influence towards therapeutic window of trifluoperazine.Ganoderic acid B has an...
TN5171 Tricetin Apoptosis , Others , Nrf2
Tricetin is a flavonoid isolated from pomegranate.Tricetin is a potent competitive inhibitor of Keap1-Nrf2 protein-protein interaction (PPI) and protects Parkinson's disease patients from 6-OHDA-induced neurotoxicity by ...
T5S0983 Absinthin Absinthiin,Absynthin HIV Protease
Absinthin (Absynthin) is a weak HIV-1 protease inhibitor.
TN4347 Jacoumaric acid HIV Protease
Jacoumaric acid is a lead molecule from the library or database of natural compounds as a HIV-1 protease inhibitor.
T10928 Cytochalasin A HIV Protease
Cytochalasin A is a cell-permeable fungal toxin and is an oxidized derivative of cytochalasin B. Cytochalasin A is an inhibitor of HIV-1 protease (IC50 = 3 μM), inhibits actin polymerization and interferes with microtubu...
T73900 (±)-Alliin
(±)-Alliin, the principal active component in garlic, functions as a potential inhibitor of SARS-CoV-2's main protease (Mpro) [1].
T79947 10-Hydroxyaloin A SARS-CoV
Hydroxyaloin A (10-10-Hydroxyaloin A) is a potent inhibitor of SARS-CoV-2, demonstrating significant efficacy in binding to the active site of the SARS-CoV-2 main protease (M^pro) [1].
T75648 Rivulariapeptolides 1155
Rivulariapeptolides 1155 is a potent serine protease inhibitor, exhibiting inhibitory concentrations (IC50s) of 41.84 nM, 4.94 nM, and 56.54 nM against chymotrypsin, elastase, and proteinase K, respectively [1].
T75649 Rivulariapeptolides 1185
Rivulariapeptolides 1185, a highly potent and selective serine protease inhibitor, exhibits IC50 values of 13.17 nM for chymotrypsin, 23.59 nM for elastase, and 55.26 nM for proteinase K [1].
T75651 Rivulariapeptolides 988
Rivulariapeptolides 988 demonstrates significant potency and selectivity as a serine protease inhibitor, exhibiting IC50 values of 95.46 nM for chymotrypsin, 15.29 nM for elastase, and 85.50 nM for proteinase K [1].
T75650 Rivulariapeptolides 1121
Rivulariapeptolides 1121 is a potent and selective serine protease inhibitor, demonstrating IC50 values of 35.52 nM for chymotrypsin, 13.24 nM for elastase, and 48.05 nM for proteinase K [1].
T75652 Molassamide B
Molassamide B, a serine protease inhibitor, exhibits potent inhibitory activity, as evidenced by its IC50 values of 24.65 nM against chymotrypsin, 11.69 nM against elastase, and 5.42 nM against proteinase K [1].
T72508 Palmatine hydroxide
Palmatine hydroxide is an orally active, irreversible inhibitor of indoleamine 2,3-dioxygenase 1 (IDO-1), demonstrating IC50 values of 3 μM for HEK 293-hIDO-1 and 157μM for rhIDO-1. Additionally, it uncompetitively inhib...

Natural Products

Hinokiflavone
T4S0181
Synonym:
Target: MMP, BCL, E1/E2/E3 Enzyme
Ganoderic acid B
TN1059
Synonym:
Target: IL Receptor, HIV Protease, JAK, STAT
Tricetin
TN5171
Synonym:
Target: Apoptosis, Others, Nrf2
Absinthin
T5S0983
Synonym: Absinthiin,Absynthin
Target: HIV Protease
Jacoumaric acid
TN4347
Synonym:
Target: HIV Protease
Cytochalasin A
T10928
Synonym:
Target: HIV Protease
(±)-Alliin
T73900
Synonym:
Target:
10-Hydroxyaloin A
T79947
Synonym:
Target: SARS-CoV
Rivulariapeptolides 1155
T75648
Synonym:
Target:
Rivulariapeptolides 1185
T75649
Synonym:
Target:
Rivulariapeptolides 988
T75651
Synonym:
Target:
Rivulariapeptolides 1121
T75650
Synonym:
Target:
Molassamide B
T75652
Synonym:
Target:
Palmatine hydroxide
T72508
Synonym:
Target:

Recombinant Proteins

Species：
Human (1567)
Mouse (231)
Cynomolgus (25)
Rat (25)
Chinese hamster (4)
Human & Mouse (4)
Human,Cynomolgus,Rhesus (4)
RSV (4)
Phleum pratense (3)
Human,Rhesus (2)
Expression System：
HEK293 Cells (1452)
E. coli (220)
Baculovirus Insect Cells (188)
CHO Cells (14)
P. pastoris (Yeast) (10)
Tag：
His (383)
C-His (333)
C-His-Avi (316)
C-hFc (202)
N-His (113)
Tag Free (111)
His, GST (75)
hFc (59)
C-mFc (40)
His, Avi (39)
Cat No. Product Name Species Expression System
TMPJ-00505 Serpin A1 Protein, Human, Recombinant (aa 25-418, His) Human HEK293 Cells
Serpin A1 is a prototype member of the Serpin superfamily of the serine protease inhibitors. As one of the most abundant proteinase inhibitors in the circulation, it is synthesized in hepatocytes, and to a lesser extent,...
TMPJ-01069 Serpin A1e Protein, Mouse, Recombinant (His) Mouse HEK293 Cells
Alpha-1-antitrypsin 1-5(SERPIN A1) is a secreted protein and belongs to the serpin family. Serpins bind the protease active site resulting in a major conformational rearrangement that traps the enzyme in a covalent acyl-...
TMPY-01589 Serpin B10 Protein, Mouse, Recombinant (His) Mouse Baculovirus Insect Cells
Serpins are the largest and most diverse family of serine protease inhibitors which are involved in a number of fundamental biological processes such as blood coagulation, complement activation, fibrinolysis, angiogenesi...
TMPK-00195 TFPI Protein, Human, Recombinant (His & Avi), Biotinylated Human HEK293 Cells
Oestrogens influence the pathophysiology and development of hormone-sensitive cancers, such as breast cancer. Tissue factor pathway inhibitor (TFPI) is a serine protease inhibitor of the extrinsic coagulation pathway and...
TMPK-00194 TFPI Protein, Human, Recombinant (His & Avi) Human HEK293 Cells
Oestrogens influence the pathophysiology and development of hormone-sensitive cancers, such as breast cancer. Tissue factor pathway inhibitor (TFPI) is a serine protease inhibitor of the extrinsic coagulation pathway and...
TMPY-01855 Serpin A10 Protein, Mouse, Recombinant (His) Mouse HEK293 Cells
Protein Z-dependent protease inhibitor, also known as PZ-dependent protease inhibitor, SERPINA1 and ZPI, is a secreted protein that belongs to the serpin family. It is expressed by the liver and secreted in plasma. SERPI...
TMPJ-01032 SPINK7 Protein, Human, Recombinant (His) Human HEK293 Cells
Serine protease inhibitor Kazal-type 7(SPINK7) is a secreted protein, that in humans is encoded by the SPINK7 gene. SPINK7 contains 1 Kazal-like domain. SPINK7 is probably serine protease inhibitor. Recombinant human SPI...
TMPJ-00625 Serpin E1 Protein, Mouse, Recombinant (His) Mouse HEK293 Cells
Plasminogen activator inhibitor-1 (serpin E1) is a serine protease inhibitor which belongs to the serpin family. Serpin E1 acts as 'bait' for tissue plasminogen activator, urokinase, protein C and matriptase-3/TMPRSS7. I...
TMPY-01841 Serpin I2 Protein, Human, Recombinant (His) Human HEK293 Cells
Serpins are the largest and most diverse family of serine protease inhibitors which are involved in some fundamental biological processes such as blood coagulation, complement activation, fibrinolysis, angiogenesis, infl...
TMPY-01814 GASP-1/WFIKKN2 Protein, Human, Recombinant (His) Human HEK293 Cells
WAP, kazal, immunoglobulin, kunitz and NTR domain-containing protein 2, also known as Growth and differentiation factor-associated serum protein 1, WAP, follistatin, immunoglobulin, kunitz and NTR domain-containing-relat...
TMPJ-00025 CST7 Protein, Human, Recombinant (His) Human HEK293 Cells
CST7 is a secreted protein and primarily expressed in peripheral blood cells and spleen.It is belongs to the cystatin family. The cystatin superfamily encompasses proteins that contain multiple cystatin-like sequences. S...
TMPY-02070 Cystatin SN Protein, Human, Recombinant (His) Human HEK293 Cells
Cystatin-SN, also known as Cystain-SA-I, Cystatin-1, Salivary cystatin-SA-1 and CST1, is a secreted protein which belongs to thecystatin family. The cystatin superfamily encompasses proteins that contain multiple cyst...
TMPY-01632 Serpin B4 Protein, Mouse, Recombinant (His) Mouse Baculovirus Insect Cells
Serpins are the largest and most diverse family of serine protease inhibitors which are involved in a number of fundamental biological processes such as blood coagulation, complement activation, fibrinolysis, angiogenesi...
TMPJ-00891 Kallikrein 2/KLK2 Protein, Human, Recombinant (His) Human HEK293 Cells
Kallikrein-2 (KLK2) is a secreted serine protease that belongs to the peptidase S1 family of Kallikrein subfamily. KLK2 contains 1 peptidase S1 domain. It is highly expressed in the human prostate gland. KLK2 can cleave ...
TMPJ-00733 SPINK1 Protein, Human, Recombinant (His) Human HEK293 Cells
Serine Protease Inhibitor Kazal-Type 1 (SPINK1) is a trypsin inhibitor that prevent the trypsin-catalyzed premature activation of zymogens within the pancreas. Defects in SPINK1 are a cause of pancreatitis (PCTT). A dise...
TMPY-02090 Cystatin B Protein, Human, Recombinant (His) Human E. coli
Cystatin-B, also known as CPI-B, Liver thiol proteinase inhibitor, Stefin-B, CSTB and CST6, is a cytoplasm and nucleus protein which belongs to thecystatin family. Cystatin-B / CSTB is an intracellular thiol proteinas...
TMPY-01711 Serpin B2 Protein, Human, Recombinant (GST) Human Baculovirus Insect Cells
Serpins are the largest and most diverse family of serine protease inhibitors which are involved in some fundamental biological processes such as blood coagulation, complement activation, fibrinolysis, angiogenesis, infl...
TMPY-02712 Serpin B3 Protein, Human, Recombinant (His) Human Baculovirus Insect Cells
SERPINB3, also known as SCCA-1, belongs to the serpin family. Serpins are a group of proteins with similar structures that were first identified as a set of proteins able to inhibit proteases. The acronym serpin was orig...
TMPY-01303 Serpin A3 Protein, Human, Recombinant (His) Human HEK293 Cells
SerpinA3, also known as Alpha 1-antichymotrypsin (AACT), is a plasma alpha globulin glycoprotein, and is a member of serpin superfamily of the serine protease inhibitors consisting of at least 35 members. SerpinA3 has be...
TMPY-04451 AMPK (G1/B1/A1) Heterotrimer Protein, Human, Recombinant (His & GST) Human Baculovirus Insect Cells
AMPK (G1/B1/A1) Heterotrimer Protein, Human, Recombinant (His & GST) is expressed in Baculovirus insect cells with His and GST tag. The predicted molecular weight is 160 kDa and the accession number is P54619-1&Q9Y478-1&...
TMPY-03878 Integrin alpha V beta 6 Protein, Human, Recombinant (Flag & His) Human HEK293 Cells
Integrin alpha V beta 6 Protein, Human, Recombinant (Flag & His) is expressed in HEK293 mammalian cells with Flag and His tag. The predicted molecular weight is 190.4 kDa and the accession number is P06756-1&P18564-1.
TMPY-02501 CD3D & CD3E Heterodimer Protein, Human, Recombinant Human HEK293 Cells
CD3D & CD3E Heterodimer Protein, Human, Recombinant is expressed in HEK293 mammalian cells. The predicted molecular weight is 77.5 kDa and the accession number is P04234-1&P07766-1.
TMPY-03745 CD3D & CD3E Heterodimer Protein, Human, Recombinant (Flag & His) Human HEK293 Cells
CD3D & CD3E Heterodimer Protein, Human, Recombinant (Flag & His) is expressed in HEK293 mammalian cells with Flag and His tag. The predicted molecular weight is 31.05 kDa and the accession number is P04234-1&P07766-1.
TMPY-03958 TGF alpha Protein, Human, Recombinant Human E. coli
The miR-137 served as a tumor suppressor in non-small cell lung cancer (NSCLC) and its suppressive effect is mediated by repressing TGFA expression. TGFA gene expression was significantly higher in tumor tissues compared...
TMPY-04069 Neurotrophin 3 Protein, Human, Recombinant Human E. coli
NTF3 (Neurotrophin 3) is a Protein Coding gene. The protein encoded by this gene is a member of the neurotrophin family, that controls the survival and differentiation of mammalian neurons. This protein is closely relate...
TMPY-02907 FGF-19 Protein, Human, Recombinant Human E. coli
FGF19, also known as FGF-19, is a member of the fibroblast growth factor (FGF) family. FGF family members possess broad mitogenic and cell survival activities, and are involved in a variety of biological processes, inclu...
TMPK-00383 ACE2/ACEH Protein, Human, Recombinant (His & Avi) Human HEK293 Cells
ACE2 (Angiotensin I Converting Enzyme 2) is a Protein Coding gene. Diseases associated with ACE2 include Severe Acute Respiratory Syndrome and Neurogenic Hypertension.The protein encoded by this gene belongs to the angio...
TMPY-01459 TNFR1/CD120a/TNFRSF1A Protein, Human, Recombinant (His) Human HEK293 Cells
TNFR1/CD120a/TNFRSF1A Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 22.7 kDa and the accession number is P19438-1.
TMPY-01827 CD30/TNFRSF8 Protein, Human, Recombinant (His) Human HEK293 Cells
CD30/TNFRSF8 Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 40 kDa and the accession number is P28908-1.
TMPY-01776 Carboxylesterase 2/CES2 Protein, Human, Recombinant (His) Human HEK293 Cells
Carboxylesterase 2/CES2 Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 60.4 kDa and the accession number is O00748-1.
TMPY-02019 CD59 Protein, Human, Recombinant (His) Human HEK293 Cells
CD59 Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 10.2 kDa and the accession number is P13987-1.
TMPY-01461 EMAP-II/AIMP1 Protein, Human, Recombinant (His) Human E. coli
EMAP-II/AIMP1 Protein, Human, Recombinant (His) is expressed in E. coli expression system with His tag. The predicted molecular weight is 35 kDa and the accession number is Q12904-1.
TMPY-00972 FGFR2 Protein, Human, Recombinant (His & hFc) Human HEK293 Cells
FGFR2 Protein, Human, Recombinant (His & hFc) is expressed in HEK293 mammalian cells with His and hFc tag. The predicted molecular weight is 67.6 kDa and the accession number is P21802-1.
TMPY-01104 Coagulation factor XI/F11 Protein, Human, Recombinant (His) Human HEK293 Cells
Factor XI (plasma thromboplastin antecedent) is a plasma glycoprotein, and a zymogen acting as a serine protease which participates in blood coagulation as a catalyst in the conversion of factor IX to factor IXa in the p...
TMPY-01912 Cadherin 17/CDH17 Protein, Human, Recombinant (His) Human HEK293 Cells
Cadherin 17/CDH17 Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 87 kDa and the accession number is Q12864-1.
TMPY-02031 B7-H3 Protein, Human, Recombinant (His) Human HEK293 Cells
B7-H3 Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 48 kDa and the accession number is Q5ZPR3-1.
TMPY-02525 RGMA Protein, Human, Recombinant (His) Human HEK293 Cells
RGMa, also known as RGM domain family, member A, belongs to the RGM (repulsive guidance molecule) family whose members are membrane-associated glycoprotein. RGMa is a glycosylphosphatidylinositol-anchored glycoprotein th...
TMPY-04262 B7-H3 Protein, Human, Recombinant (His), Biotinylated Human HEK293 Cells
B7-H3 Protein, Human, Recombinant (His), Biotinylated is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 48 kDa and the accession number is Q5ZPR3-1.
TMPY-00915 Serpin A1 Protein, Human, Recombinant (His) Human HEK293 Cells
Serpin A1 Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 45.7 kDa and the accession number is P01009-1.
TMPY-02836 MFGE8 Protein, Human, Recombinant (His) Human Baculovirus Insect Cells
MFGE8 Protein, Human, Recombinant (His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 42 kDa and the accession number is Q08431-1.
TMPY-01462 IL-11R alpha/IL-11RA Protein, Human, Recombinant (His) Human HEK293 Cells
IL-11R alpha/IL-11RA Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 38.6 kDa and the accession number is Q14626-1.
TMPK-00176 BAFF/TNFSF13B Trimer Protein, Human, Recombinant (His & Flag) Human HEK293 Cells
B-cell activating factor (BAFF) also known as tumor necrosis factor ligand superfamily member 13B is a protein that in humans is encoded by the TNFSF13B gene.BAFF is a cytokine that belongs to the tumor necrosis factor (...
TMPY-02034 Siglec-2/CD22 Protein, Human, Recombinant (His) Human HEK293 Cells
Siglec-2/CD22 Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 76.6 kDa and the accession number is P20273-1.
TMPY-02794 TLR2 Protein, Human, Recombinant (aa 1-587, His) Human Baculovirus Insect Cells
TLR2 Protein, Human, Recombinant (aa 1-587, His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 65.5 kDa and the accession number is O60603-1.
TMPY-04799 IFNAR2 Protein, Human, Recombinant (His), Biotinylated Human HEK293 Cells
IFNAR2 Protein, Human, Recombinant (His), Biotinylated is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 26.2 kDa and the accession number is P48551-1.
TMPY-02647 IFNAR1 Protein, Human, Recombinant (His) Human HEK293 Cells
IFNAR1 Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 48.6 kDa and the accession number is P17181-1.
TMPY-04826 LILRB5/CD85c Protein, Human, Recombinant (His) Human HEK293 Cells
A genetic variant in LILRB5 (leukocyte immunoglobulin-like receptor subfamily-B) (rs12975366: T > C: Asp247Gly) has been reported to be associated with lower creatine phosphokinase (CK) and lactate dehydrogenase (LDH) le...
TMPY-00740 SDF-1 Protein, Human, Recombinant (hFc) Human HEK293 Cells
SDF-1 Protein, Human, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 35.2 kDa and the accession number is P48061-1.
TMPY-04698 HER2/ERBB2 Protein, Human, Recombinant (aa 489-630, His) Human HEK293 Cells
HER2/ERBB2 Protein, Human, Recombinant (aa 489-630, His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 17.1 kDa and the accession number is P04626-1.
TMPY-00203 LOXL2 Protein, Mouse, Recombinant (His) Mouse HEK293 Cells
Lysyl oxidase homolog 2, also known as Lysyl oxidase-like protein 2, Lysyl oxidase-related protein 2, Lysyl oxidase-related protein WS9-14 and LOXL2, is a secreted protein that belongs to the lysyl oxidase family. LOXL2 ...
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Serpin A1 Protein, Human, Recombinant (aa 25-418, His)
TMPJ-00505
Species: Human
Expression System: HEK293 Cells
Serpin A1e Protein, Mouse, Recombinant (His)
TMPJ-01069
Species: Mouse
Expression System: HEK293 Cells
Serpin B10 Protein, Mouse, Recombinant (His)
TMPY-01589
Species: Mouse
Expression System: Baculovirus Insect Cells
TFPI Protein, Human, Recombinant (His & Avi), Biotinylated
TMPK-00195
Species: Human
Expression System: HEK293 Cells
TFPI Protein, Human, Recombinant (His & Avi)
TMPK-00194
Species: Human
Expression System: HEK293 Cells
Serpin A10 Protein, Mouse, Recombinant (His)
TMPY-01855
Species: Mouse
Expression System: HEK293 Cells
SPINK7 Protein, Human, Recombinant (His)
TMPJ-01032
Species: Human
Expression System: HEK293 Cells
Serpin E1 Protein, Mouse, Recombinant (His)
TMPJ-00625
Species: Mouse
Expression System: HEK293 Cells
Serpin I2 Protein, Human, Recombinant (His)
TMPY-01841
Species: Human
Expression System: HEK293 Cells
GASP-1/WFIKKN2 Protein, Human, Recombinant (His)
TMPY-01814
Species: Human
Expression System: HEK293 Cells
CST7 Protein, Human, Recombinant (His)
TMPJ-00025
Species: Human
Expression System: HEK293 Cells
Cystatin SN Protein, Human, Recombinant (His)
TMPY-02070
Species: Human
Expression System: HEK293 Cells
Serpin B4 Protein, Mouse, Recombinant (His)
TMPY-01632
Species: Mouse
Expression System: Baculovirus Insect Cells
Kallikrein 2/KLK2 Protein, Human, Recombinant (His)
TMPJ-00891
Species: Human
Expression System: HEK293 Cells
SPINK1 Protein, Human, Recombinant (His)
TMPJ-00733
Species: Human
Expression System: HEK293 Cells
Cystatin B Protein, Human, Recombinant (His)
TMPY-02090
Species: Human
Expression System: E. coli
Serpin B2 Protein, Human, Recombinant (GST)
TMPY-01711
Species: Human
Expression System: Baculovirus Insect Cells
Serpin B3 Protein, Human, Recombinant (His)
TMPY-02712
Species: Human
Expression System: Baculovirus Insect Cells
Serpin A3 Protein, Human, Recombinant (His)
TMPY-01303
Species: Human
Expression System: HEK293 Cells
AMPK (G1/B1/A1) Heterotrimer Protein, Human, Recombinant (His & GST)
TMPY-04451
Species: Human
Expression System: Baculovirus Insect Cells
Integrin alpha V beta 6 Protein, Human, Recombinant (Flag & His)
TMPY-03878
Species: Human
Expression System: HEK293 Cells
CD3D & CD3E Heterodimer Protein, Human, Recombinant
TMPY-02501
Species: Human
Expression System: HEK293 Cells
CD3D & CD3E Heterodimer Protein, Human, Recombinant (Flag & His)
TMPY-03745
Species: Human
Expression System: HEK293 Cells
TGF alpha Protein, Human, Recombinant
TMPY-03958
Species: Human
Expression System: E. coli
Neurotrophin 3 Protein, Human, Recombinant
TMPY-04069
Species: Human
Expression System: E. coli
FGF-19 Protein, Human, Recombinant
TMPY-02907
Species: Human
Expression System: E. coli
ACE2/ACEH Protein, Human, Recombinant (His & Avi)
TMPK-00383
Species: Human
Expression System: HEK293 Cells
TNFR1/CD120a/TNFRSF1A Protein, Human, Recombinant (His)
TMPY-01459
Species: Human
Expression System: HEK293 Cells
CD30/TNFRSF8 Protein, Human, Recombinant (His)
TMPY-01827
Species: Human
Expression System: HEK293 Cells
Carboxylesterase 2/CES2 Protein, Human, Recombinant (His)
TMPY-01776
Species: Human
Expression System: HEK293 Cells
CD59 Protein, Human, Recombinant (His)
TMPY-02019
Species: Human
Expression System: HEK293 Cells
EMAP-II/AIMP1 Protein, Human, Recombinant (His)
TMPY-01461
Species: Human
Expression System: E. coli
FGFR2 Protein, Human, Recombinant (His & hFc)
TMPY-00972
Species: Human
Expression System: HEK293 Cells
Coagulation factor XI/F11 Protein, Human, Recombinant (His)
TMPY-01104
Species: Human
Expression System: HEK293 Cells
Cadherin 17/CDH17 Protein, Human, Recombinant (His)
TMPY-01912
Species: Human
Expression System: HEK293 Cells
B7-H3 Protein, Human, Recombinant (His)
TMPY-02031
Species: Human
Expression System: HEK293 Cells
RGMA Protein, Human, Recombinant (His)
TMPY-02525
Species: Human
Expression System: HEK293 Cells
B7-H3 Protein, Human, Recombinant (His), Biotinylated
TMPY-04262
Species: Human
Expression System: HEK293 Cells
Serpin A1 Protein, Human, Recombinant (His)
TMPY-00915
Species: Human
Expression System: HEK293 Cells
MFGE8 Protein, Human, Recombinant (His)
TMPY-02836
Species: Human
Expression System: Baculovirus Insect Cells
IL-11R alpha/IL-11RA Protein, Human, Recombinant (His)
TMPY-01462
Species: Human
Expression System: HEK293 Cells
BAFF/TNFSF13B Trimer Protein, Human, Recombinant (His & Flag)
TMPK-00176
Species: Human
Expression System: HEK293 Cells
Siglec-2/CD22 Protein, Human, Recombinant (His)
TMPY-02034
Species: Human
Expression System: HEK293 Cells
TLR2 Protein, Human, Recombinant (aa 1-587, His)
TMPY-02794
Species: Human
Expression System: Baculovirus Insect Cells
IFNAR2 Protein, Human, Recombinant (His), Biotinylated
TMPY-04799
Species: Human
Expression System: HEK293 Cells
IFNAR1 Protein, Human, Recombinant (His)
TMPY-02647
Species: Human
Expression System: HEK293 Cells
LILRB5/CD85c Protein, Human, Recombinant (His)
TMPY-04826
Species: Human
Expression System: HEK293 Cells
SDF-1 Protein, Human, Recombinant (hFc)
TMPY-00740
Species: Human
Expression System: HEK293 Cells
HER2/ERBB2 Protein, Human, Recombinant (aa 489-630, His)
TMPY-04698
Species: Human
Expression System: HEK293 Cells
LOXL2 Protein, Mouse, Recombinant (His)
TMPY-00203
Species: Mouse
Expression System: HEK293 Cells
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Cat No. Product Name
L1100 Protease Inhibitor Library

343 compounds
A unique collection of 343 protease and proteasome inhibitors for research in chemical genomics, and drug screening;

Libraries

Protease Inhibitor Library
L1100
Compounds: 343

Reagents


RIPA Lysis Buffer
(Strong)
Catalog No. C0045
RIPA Lysis Buffer
(Middle)
Catalog No. C0046
RIPA Lysis Buffer
(Weak)
Catalog No. C0047
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